Ever since its discovery and availability for sale and use in the late 1940s, lidocaine has become an exceptionally commonly used medication [T583]. In particular, lidocaine's principal mode of action in acting as a local anesthetic that numbs the sensations of tissues means the agent is indicated for facilitating local anesthesia for a large variety of surgical procedures [F4349, L5930, L5948]. It ultimately elicits its numbing activity by blocking sodium channels so that the neurons of local tissues that have the medication applied on are transiently incapable of signaling the brain regarding sensations [F4349, L5930, L5948]. In doing so, however, it can block or decrease muscle contractile, resulting in effects like vasodilation, hypotension, and irregular heart rate, among others [F4349, L5930, L5948]. As a result, lidocaine is also considered a class Ib anti-arrhythmic agent [L5930, L5948, F4468]. Nevertheless, lidocaine's local anesthetic action sees its use in many medical situations or circumstances that may benefit from its action, including the treatment of premature ejaculation [A177625]. Regardless, lidocaine is currently available as a relatively non-expensive generic medication that is written for in millions of prescriptions internationally on a yearly basis. It is even included in the World Health Organization's List of Essential Medicines [L6055].
Synonyms
2-(Diethylamino)-N-(2,6-dimethylphenyl)acetamide
Lignocaine
Lidocaine
Lidoca¨ªna
¦Á-diethylamino-2,6-dimethylacetanilide
alpha-diethylamino-2,6-dimethylacetanilide
Lidocaine hydrochloride anhydrous
Lidocainum
2-(Diethylamino)-2',6'-acetoxylidide
Lidocaine hydrochloride
Lidocaina
Brand Names
Small Cuts and Burns
TopCare Pain Relieving Analgesic
Preparation H Rapid Relief
GENUINE FIRST AID Emergency Preparedness Contains 167 PIECES HARDCASE
Lidotral 3.88% Roll on
DG Health Pain Relieving
Afassco First Aid Burn Cream
Numb Soothe
Hemorrhoid Relief Cream
Antibiotic Cream Plus Pain Relief
Seaford Nifedipine and Lidocaine Hydrochloride Cream
ACTIVE-PAC with Gabapentin
AnaMantle HC
Lidocare 03
Burn Treatment
Disposable Convenience Kit (Single Shot Epidural)
NUMB PLUS Maximum Strength Anorectal
4254 First Aid Kit
4375 First Aid Kit
Doloracin/l Rx With Lidocaine
4308 First Aid Kit
Jamshidi Bone Marrow Biopsy Tray
4390 First Aid Kit
Sore relief
Hempvana Knee Bird Ultra Strength Pain Relief
Bottoms Up Health
CVS Health Lidocaine Pain Relief Plus Menthol
Lidocaine Ont 5% Graham Flavored
DG health
Lido Rx
Yowch for minor burns by Pain Balm
4187 First Aid Kit
Harmony Products LLC.
Lidocaine with Menthol
Genuine First Aid Industrial First Aid
4191 First Aid Kit
Apr15
Derma Gel Relief
Lidodan Cream 5%
Lidenza Patch
Hot and Cold Cream with Lidocaine Pain Relieving
Walgreens Cooling
Equate Hemorrhoid Relief
biochemistry PAIN RELIEF FOOT ACTIVE
DermacinRx DPN Pak
UniShield First Aid Burn
4273 First Aid Kit
Walgreens
ARC FIRST AID Contains 101 PIECES Hardcase
Lidocaine Hydrochloride Injection, USP 1%
Tylenol Precise Pain Relieving
4206 First Aid Kit
4086 First Aid Kit
Walgreens Burn
Rite Aid Rectal Care
Dexlido-M Kit
Australian Gold Aloe Freeze Gel with Lidocaine
Lidopen
Ketorocaine LM Kit
4248 First Aid Kit
Lidodan 4% Topical Solution
Lidocaine 2% and Epinephrine 1:50 000
Relyyks
First Aid Antiseptic Well at Walgreens
Truu Balance Pain Relief
Premium Lidocaine
Burn Relief Aloe Vera Gel GNP
Soundbody
Extra Strength AfterTAT Slime
Fast Freeze Lidocaine Roll-On
4397 First Aid Kit
Doctor Butler Hemorrhoid and Fissure Advanced Formula
ABSORBINE jr.
Bikini Relief
Zee Burn Relief
Comfortcaine
Base Numb Topical Anorectal
Lidopatch
SYREN Intimate Relief Topical Pain Relief
CBD PAIN RELIEF Cream
LidAll
BeKoool Itch Relief
Ozonol Antibiotic Plus - Ointment
Zovacil 5
Walgreens Lidocaine Plus Cream
Lidocaine Hydrochloride Injection
Bed Bug Instant Bite Relief
Footworks Maximum Strength Cracked Heel
4104 First Aid Kit
Pharmacist Choice TSX Transdermal Patch
ACT Kit (Accelerated COVID-19 Test Kit)
LidoReal-30 4% Topical Patch
4379 First Aid Kit
Fruit of the Earth Cool Blue Aloe Mist Continuous
Hemorrhoid Relief
Vallement Flex
Extra Strength Numbing Gel
Xylocaine 2% With Epinephrine 1:200000
Walgreens pain relieving
QKit Procedure Tray
Lidocaine Hci and Epinephrine
Multi-Specialty Kit
PRILOVIX Ultralite Plus
Caribbean Breeze Burn Relief
Steady Freddy
Xylocaine Mpf
Pain Relieving Lidocaine Patch
Atozcup Tattoo Numbing
Hemorrhoid and Fissure Dr. Butler
Super-Stop BloodClotter
4261 First Aid Kit
Solarcaine First Aid Lidocaine Spray
Stud 100
Diclovix
Meijer Lidocaine Pain Relief Patch Assortment Medium
Octocaine HCl 2% Epinephrine 1:100000
First Aid Kit 64058024
Prilovix
Lido-mp40
Extra Strength AfterTAT
ECOLAB Blood Clotting
Lidocaine 3% Topical Anesthetic Cream
Re-Lieved Lidocaine Patch
First Aid and Burn
H-Releve Hemorrhoidal
Atelocollagen Implant
Electrum Numb Foam
Preginot
Lidocaine Dry Patch Plus Menthol
Lidodan Viscous 2%
Sinsinpas Lidocaine Pain Relieving
Rugby PAIN RELIEF PATCHES
Inflammation Reduction Pack
Lipritin
Premjact Male Desensitizer Pound International
MEDI-FIRST Topical Analgesic
Holy Water Mercy In A Bottle
AOBBIY Tattoo Numbing Cream
4389 First Aid Kit
4373 First Aid Kit
Bactine Max Dry
Ebsl-5
Odynia-UUltra Patch Ultra Patch
4115 First Aid Kit
Walgreens 24-Hour Lidocaine Patch
Absorbine Jr Pro Cream
Lidovex
4 Lidocaine Topical Anesthetic
ReadySharp Anesthetics plus Ketorolac
Lidolog Kit
4192 First Aid Kit
Realheal-I
ScleraCare Lidocaine HCL
Limencin
MLK Kit F2
Zylotrol Plus
Lidothol Gel
AUVON LIDOCAINE MENTHOL Pain Relief
Lidocaine Hydrochloride Gel
QC Lidocaine Maximum Strength
Lidopro
Rematex
Restoriden Lidocaine Cream
Dermatool Hemorrhoidal
50 Person ANSI
MyDerm
PainPatrol CBD Pain Relief with Lidocaine
CBD Pain
LM Plus Relief
Footworks Healthy Cracked Heel Cream
Xylocaine 0.5% W Epinephrine 1:200000
Lido-RX 4.1
Hot and Cold with Lidocaine Pain Relieving
Zee First Aid Cream
Lidopin
Dyural 80-LM
Cathejell
Ritual Tattoo
Rapid Pain-relief Topical
4222 First Aid Kit
Elite PAIN RELIEF
Leader Lidocaine
D-Care 100X
Easy Care First Aid Kit - Comprehensive
LevigoSP
Xpacaine
ReCellTis Wound Cream
Tpr20
ARC Emergency Preparedness FIRST AID Contains 202 PIECES
Prelidopine Pre-Operative System
Walgreens Cool N Heat Dry
Pain Relief Lidocaine
Aloe Gel Pain Reliever Well at Walgreens
ARC FIRST AID Emergency Preparedness Contains 167 PIECES
Point Of Care L5
Inkeeze Original B Numb Cylinder
Panama Jack Burn Relief Gel with Lidocaine
Topicaine 5
4301 First Aid Kit
Extra Strength Naturally Hl Sunburn Relief
Greencaine Blast
Tidl Pain Relief Numbing Tidl
Dolotranz
Meijer Burn Relief Aloe Vera Pain Relieving Gel
Medi-First Plus Burn with Lidocaine
Burn with Aloe
4395 First Aid Kit
Pain Relieving Gel-Patch
RadiaGuard Advanced Radiation Relief
First Aid Antiseptic Rite Aid pharmacy
Safetec Burn Spray
CANNA NUMB Roll On
4347 First Aid Kit
Lidocaine 2% and Epinephrine 1:50,000
Sj3
Fruit of the Earth Aloe Vera Cool Blue
Alocane On The Go
Maximum Strenght Lidocaine plus Menthol Pain Relief Patch
Pre-wax Pain Relief
Absorbine jr. Lidocaine
Botanika Life Soothing Pain Serum
CLIN-LIDO-Single Use Kit
GoodSense Pain Relief
Numb 100
Medicated Pain Relief Foot CVS
EZ-Relief
Naturally HL Extra Strength Insect Bite Numbing
Prilo Patch-II
4052 First Aid Kit
Assured Bikini Smooth Cream
CVS Health XL Lidocaine Pain Relief
Hempvana Maximum Strength Pain Relief Cream
Zcaine Fast Acting Anesthetic
First Aid Antiseptic Pain Relieving Cream
Alcoholada Gel Pain Relieving Pain
NATURES CRAFT LIDOCAINE Male Genital Desensitizer
Painless Tattoo 2
4064 First Aid Kit
Precise Cooling Pain Relief Cream
Pantin
Bufferin Lidocaine Pain Numbing
Mld
Ritual Tattoo Reveal Foam
4148 First Aid Kit
Physician EZ Use Joint Tunnel and Trigger Kit II
Zylotrol Pain Relieving
Trifena
Gardeners Skin Remedy Topical Analgesic Gel
Hyronan
Lidocan IV
WPR Plus
Leader
Lipsorex Plus
Nanonumb
4099 First Aid Kit
4342 First Aid Kit
Lidocaine 2% and Epinephrine 1:100,000
Polysporin Complete
Aspercreme with Lidocaine
Inderma MD
Pro-C-Dure 4 Kit
Topical Pain Relief
DermaNumb Anesthetic Gel
DYNAMO DELAY Black Label
Blackwork
FourPainRX
MAXOCAINE Lidocaine Hemp Oil Topical Analgesic
Kendra SKIN PROTECTION and PAIN RELIEF FOR HAIR REMOVAL
4184 First Aid Kit
Hempvana Ultra Strength Pain Relief Cream
Numbing Label
CBD Pain Patches
Toplast Pain Relief Lidocaine 4percent
VacuStim Silver
Anecream
Topicaine
Aramark Burn
Triderma Pain Relief
Zilacaine Patch
4045 First Aid Kit
Burn Relief Professional Bio-Kool
Numbing Hemorrhoidal Label
Prikaan Lite
4007 First Aid Kit
Curist Lidocaine Maximum Strength
4032 First Aid Kit
4153 First Aid Kit
Lidocaine 4 Percent PLUS
Skin Soothing Aid
Numb Master
Alcoholada Pain Relieving
4098 First Aid Kit
Coralite Lidocaine Pain Relief
Numquick Topical Analgesic
Penichillin
Lidocaine 4 Percent and Menthol 1 Percent Roll-On
Solarcaine
Lidovix Delayed Release
4196 First Aid Kit
Aloe
Pro Numb
Recticare
Lidocaine-Prilocaine-Cream Base
Emla
4111 First Aid Kit
Res-Q Topical Analgesic Soothing Gel
Pain Relief Roll-on Good Sense
BonaDur
Nupharmisto Tattoo Numbing Cream
Gold Bond Medicated Pain and Itch Relief
Lidozo Topical Pain Patch
Lidocaine 4%
Lidotin
CVS Burn Relief w/Lido 8oz
Dyural LM Kit
Lidocaine Menthol Pain Relief
XYLOCAINE- MPF (LIDOCAINE HCl )
BLUE ACME SLEEVE FIRST AID Contains 1000 PIECES
Lidocan
Family Medic First-aid Treatment Lotion
Icy Hot with Lidocaine Pain Relieving
Lidotral 3.88 Percent Plus Hydrocortisone 1 Percent
Ocean Breeze Pain Relief
Siterol
Duloxicaine
4345 First Aid Kit
LidoHeal-90
Leximenth
4132 First Aid Kit
BZ Step Pain Relief Cream
Wound Debridement Kit
Terrasil Cold Sore Treatment Max
Myelogram Tray 1%
ReadySharp Anesthetics plus Dexamethasone
Polysporin Plus Pain Relief
Natural Seal Itch Relief for Kids
Cyclopak
Good Neighbor Pharmacy Emergency Preparedness and First Aid Contains 167 Pieces
Pure-Aid
GFA First Aid 16 Unit Metal Case
Base Laboratories Base Numb Topical Anorectal Cream
Extra Strength Naturally HL Warming Ice
PAIN RELIEF Gel-Roll On
Extra Strength Shingles Chickenpox Relief
Xylocaine Co2 Inj
4150 First Aid Kit
ReadySharp-P40
Sunburn Relief
Alocane Emergency Burn
4270 First Aid Kit
Lidocaine Patch
LIDOCAINE PAIN RELIEF Gel-Patch
CVSLidocaineAntisepticSpray
4326 First Aid Kit
Lidocaine 2% and Epinephrine 1:100 000
Signature Care Lidocaine Cream
CVS Health Maximum Strength Lidocaine Pain Relief Cream Plus Menthol
First Shield
Burn Relief Signature Care
First Aid Burn
DermacinRx Prizopak
4116 First Aid Kit
4352 First Aid Kit
Lidocaine Hydrochloride and 5% Dextrose Injection USP
Jampocaine 2% Viscous Solution
Dzul - Lido Creme Maximum Strength
4372 First Aid Kit
Lidonex
Fossaoprin SPG2
DCH Pain Relief
Aramark Blood Clotting
Sunburn Pain relief
Zionodil 50
Lidocoll
Lidocaine HCl Inj 1%
4110 First Aid Kit
Xylocaine 1.5%
Hydrocaine
First Aid Triple Antibiotic with Pain Reliever
Tridacaine XL
Afassco Burn Gel
Burn Ease
Crane Safety Burn
Premier Value Pain Relief Patches
Lyracaine Gel
BENGAY Tropical Jasmine
Salonpas Pain Relieving LIDOCAINE 4% FLEX
NOpioid-TC
Jamshidi Menghini Soft Tissue Biopsy Tray
Minnerva II
American Safety First Aid
Lidocaine HCl and Hydrocortisone Acetate
2677 First Aid Burn Cream
Lipritin II
Swiss Navy Endurance Rx Pro
Veltrix
Dr. Richs Numbing
Base Laboratories Base Numb Extra Strength Topical Anorectal
Fsk-5
4105 First Aid Kit
Pain free IV
Calm and Correct Serum with Lidocaine
First Aid Pocket Pack - 40 Pieces
Yowch extra strength for insect bites and stings
Lidosporin Ear Drops
Remaxazon External Patch
Lidocaine Pain Relieving
Livixil Pak
Swiss Navy EnduranceRx
OKeeffes Healthy Feet
4228 First Aid Kit
Maximum Stremgth Pain Relief Good Sense
MLK F3 Kit
CVS Health Aftersun Aloe Vera Cooling
Lidovin
4253 First Aid Kit
4333 First Aid Kit
Duane Reade Aloe Vera Pain Relieving
Careland Lidocaine 4 Plus Menthol Pain Relieving Gel Patches for back, neck shoulders knees and elbows with border
LIDOCAINE HCl
Gigi Anesthetic Numbing
NORTH Antiseptic First Aid
Ocean Potion Instant Burn Relief Ice
Workvie
Analgesic
ReadySharp-P80
Lidocaine HCl Injection USP 1% (50mg/5ml)
Antiseptic Formula Filled Swab
Instant Burn Relief Aloe Extra CVS
Liprotek
P-Care K40MX
Aspercreme with Lidocaine Essential Oils Rosemary Mint
Skullduggery Pain Relief and Skin Protection for Tattoos
Burn Relief Gel
Burn Ease, 3.5g
CVS Health All Purpose Kit
Lidocaine and Epinephrine Inj.usp 2% 1:100000
After Cuts and Scrapes
Yowch Extra Strength for minor burns
4378 First Aid Kit
HealthWise Lidocaine and Menthol Pain Relief
GFA First Aid 36 Unit Metal Case
Phenyl-Lido
Exigence One Patch
4281 First Aid Kit
4359 First Aid Kit
Extra Strength Wound Care
Pain Relief 4% Lidocaine
Soothee Patch
Will Relieve
Xylocaine Mpf 1.5% With Epinephrine
Lmx5
MAKESENSE First Aid
Foot Works Healthy Cracked Heel Cream
4234 First Aid Kit
Extra Strength Foot Care Liquid Gel
Sportcaine Patch
Lidocaine Hydrochloride Topical Solution USP
1st RELIEF TOPICAL
Nuvakaan II
LifeStyles EPIC Male Genital Desensitizer
Moshe Numbing Hemorrhoidal
Foster and Thrive
CLM Patch
4322 First Aid Kit
Poly-Prep
Xylocaine -MPF
Sore Relief
Lignospan Standard
PharmapureRx Menthotral
4360 First Aid Kit
I.C.E. Lidocaine Gel - Gel Lidocaine
Medline
4310 First Aid Kit
Plush anesthetics L
Feel Better Now
Stama Pro
Burn Relief Kol-Down
Renuu Patch
4330 First Aid Kit
Pro Comfort 8 Hours Patch
GeriGentle FrostyHeat Pain Relief Patch 4 Lodocaine Back
Prizotral
Lidotral Two Percent
Sky Wellness Max Pain Relief
Xylocaine 0.5%
Numstick
Tridacaine II
Xylocaine 1.5% W Epinephrine 1:200000 Test Dose
Zone 2
4202 First Aid Kit
EPIC Burn Cream
Neptune Ice Patch
4335 First Aid Kit
Lidocaine HCl Hydrocortisone Acetate
Xylocaine Dental Lidocaine HCl 2% and Epinephrine 1:100,000
Moxicaine kit
Keepan A
LidoPure Patch
Octocaine 100 Needleject Inj
Prilovixil
Priloxx LP External Kit
Lido Pain Relief
Walgreens Pain Relieving with Turmeric Analgesic
Xylocaine-mpf, 2%
EmReal
HemRid Anorectal Cream
4376 First Aid Kit
Leader After Sun Cooling
Lidotral Five Percent
Polysporin for Stitches
4264 First Aid Kit
LexiLido
Walgreens Sunburn Relief
4338 First Aid Kit
Point Relief LidoSpot
Pain Relief Cream
Formula 4 Pain
Rugby Lidocaine
Lipovite
4280 First Aid Kit
POWERECT Max Power Male Delay
4257 First Aid Kit
Scalpanumb
ADVANCED NUMB Topical Anesthetic
Salonpas LIDOCAINE Pain Relieving
GelAzul Roll-On
Harmony Hemp NeuroComfort Pain Relief Spray500
TheraCare Pain Relief Lidocaine
Indication
Lidocaine is an anesthetic of the amide group indicated for production of local or regional anesthesia by infiltration techniques such as percutaneous injection and intravenous regional anesthesia by peripheral nerve block techniques such as brachial plexus and intercostal and by central neural techniques such as lumbar and caudal epidural blocks [F4349, L5930].
Categories
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical Use
Agents that reduce seizure threshold
Amides
Amines
Analgesics and Anesthetics
Anesthetics
Anesthetics for Topical Use
Anesthetics, Local
Anilides
Aniline Compounds
Antiarrhythmic agents
Antiarrhythmics, Class I
Antiarrhythmics, Class Ib
Antipruritics and Local Anesthetics
Antipruritics, Incl. Antihistamines, Anesthetics, Etc.
Drug Info/Drug Targets: DrugBank 3.0: a comprehensive resource for 'omics' research on drugs. Knox C, Law V, Jewison
T, Liu P, Ly S, Frolkis A, Pon A, Banco K, Mak C, Neveu V, Djoumbou Y, Eisner R, Guo AC, Wishart DS.
Nucleic Acids Res. 2011 Jan; 39 (Database issue):D1035-41. | PMID:21059682